
(43)22.05.2002 (87)en
(24) 18.01.2006
(30)25.08.1999 JP 23900499
(54) ISOINDOLDERIVATE
(73)BANYU PHARMACEUTICAL CO., LTD.
2-3, Nihombashi Honcho 2-chome
Chuo-ku, Tokyo 103-8416 (JP)
(72)NAGASE, Toshio, Banyu Pharmaceutical Co., Ltd.
Tsukuba Research Institute, 3, Okubo
Tsukuba-shi, Ibaraki 300-2611 (JP)
IINO, Tomoharu, Banyu Pharmaceutical Co., Ltd.
Tsukuba Research Institute, 3, Okubo
Tsukuba-shi, Ibaraki 300-2611 (JP)
SATO, Yoshiyuki, Banyu Pharmaceutical Co., Ltd.
Tsukuba Research Institute, 3, Okubo
Tsukuba-shi, Ibaraki 300-2611 (JP)
NISHIMURA, Teruyuki, Banyu Pharmaceutical Co.
Ltd.
Tsukuba Research Institute, 3, Okubo
Tsukuba-shi, Ibaraki 300-2611 (JP)
EIKI, Jun-ichi, Banyu Pharmaceutical Co., Ltd.
Tsukuba Research Institute, 3, Okubo
Tsukuba-shi, Ibaraki 300-2611 (JP)
(86)PCT/JP 2000/005723 (ja)
(87)WO 2001/014386 1.3.2001
(51) C 07 D 0491/10 (2006.01) Z C 07 D 0401/14 (2006.01)
(11) 01 235 825
(51) C 07 D 0491/147 (2006.01) Z C 07 D 0491/048 (2006.01)
(11) 01 207 161
(51) C 07 D 0498/04 (2006.01) Z C 07 D 0491/048 (2006.01)
(11) 01 207 161
(51) C07 D0498/04 (2006.01)
C07 D0471/04 (2006.01)
A61K0031/4741 (2006.01)
A61K0031/4745 (2006.01)
A61P0035/00 (2006.01)
C07 D0498/04 (2006.01)
C07 D0261/00 (2006.01)
C07 D0221/00 (2006.01)
C07 D0471/04 (2006.01)
C07 D0231/00 (2006.01)
C07 D0221/00 (2006.01)
C07 D0498/04 (2006.01)
C07 D0263/00 (2006.01)
C07 D0221/00 (2006.01)
(51) C 07 D 0498/04 (2006.01) Z C 07 D 0498/04 (2006.01)
(11) 01 224 189
(21) 00968314.5
(22)22.09.2000 (86)en
(43)24.07.2002 (87)en
(24) 25.01.2006
(30)07.10.1999 US 158175 P
09.12.1999 US 169784 P
(54) KONDENSIERTE DIHYDROCHINOLINON-DERIVATE
ZUR HEMMUNG VON MRP1
(73)ELI LILLY AND COMPANY
Lilly Corporate Center
Indianapolis, Indiana 46285 (US)
(72)LOHMAN, Mark, Christopher
3455 Table Mesa Drive Apartm. H-180
Boulder, CO 80305 (US)
VEPACHEDU, Sreenivasarao
16 West 630 Mockingbird Lane, Apartment 20G
Hinsdale, IL 60521 (US)
XIE, Yongping
19 Huntington Circle, Apartment 15
Naperville, IL 60540 (US)
BONJOUKLIAN, Rosanne
318 Dominion Drive
Zionsville, IN 46077 (US)
JOHNSON, Douglas, Webb
235 Saddlebrook Court
Zionsville, IN 46077 (US)
LANDER, Peter, Ambrose
5407 North Capitol Avenue
Indianapolis, IN 46208 (US)
PATEL, Vinod, Francis
3 Mossy Lane, Bellows Farm
Acton, MA 01720 (US)
(86)PCT/US 2000/021980 (en)
(87)WO 2001/027116 19.4.2001
(51) C 07 D 0498/14 (2006.01) Z C 07 D 0491/048 (2006.01)
(11) 00 697 872
(51) C 07 F 0009/40 (2006.01) Z A 61 K 0031/44 (2006.01)
(11) 00 697 872
(51) C 07 F 0009/46 (2006.01) Z B 01 J 0031/18 (2006.01)
(11) 01 446 224
(51) C 07 F 0009/48 (2006.01) Z C 07 F 0007/18 (2006.01)
(11) 01 097 158
(51) C 07 F 0009/50 (2006.01) Z C 07 F 0007/18 (2006.01)
(11) 01 097 158
(51) C 07 F 0009/547 (2006.01) Z B 01 J 0031/18 (2006.01)
(11) 01 446 224
(51) C 07 F 0009/572 (2006.01) Z C 07 F 0007/18 (2006.01)
(11) 01 097 158
(51) C 07 F 0009/58 (2006.01) Z B 01 J 0031/18 (2006.01)
(11)
01 446 224
(51) C 07 F 0009/60 (2006.01) Z B 01 J 0031/18 (2006.01)
(11) 01 446 224
(51) C 07 F 0009/6512 (2006.01) Z B 01 J 0031/18 (2006.01)
(11) 01 446 224
(51) C 07 F 0009/653 (2006.01) Z C 07 F 0007/18 (2006.01)
(11) 01 097 158
(51) C 07 F 0009/6547 (2006.01) Z C 07 F 0007/18 (2006.01)
(11) 01 097 158
(51) C 07 F 0009/6558 (2006.01) Z B 01 J 0031/18 (2006.01)
(11) 01 446 224
(51) C 07 F 0009/6571 (2006.01) Z C 07 F 0007/18 (2006.01)
(11) 01 097 158
(51) C07 F0009/6584 (2006.01)
A61K0031/675 (2006.01)
A61P0029/00 (2006.01)
A61P0019/00 (2006.01)
A61P0035/00 (2006.01)
(11) 01 470 138
(21) 03702358.7
(22)15.01.2003 (86)en
(43)27.10.2004(87)en
(24) 18.01.2006
(30)18.01.2002 US 349229 P
(54) MMP-INHIBITOREN
(73)LEO PHARMA A/S
Industriparken 55
2750 Ballerup (DK)
(72)CHRISTENSEN, Mette, Knak
Kollemosevej 33 F, 1.
DK-2840 Holte (DK)
BLAEHR, Lars, Kristian, Albert
Steen Billes Gade 1, 4.th
DK-2100 Kobenhavn (DK)
(86)PCT/DK 2003/000025 (en)
(87)WO 2003/059921 24.7.2003
(51) C 07 F 0015/00 (2006.01) Z B 01 J 0031/18 (2006.01)
(11) 01 446 224
(51) C 07 F 0015/00 (2006.01) Z C 07 F 0007/18 (2006.01)
(11) 01 097 158
(51) C 07 F 0015/04 (2006.01) Z B 01 J 0031/18 (2006.01)
(11)
01 446 224
(51) C07 F0015/06 (2006.01)
(11) 01 323 725
(21) 02028775.1
(22)23.12.2002 (86)de
(43)02.07.2003 (87)de
(24) 18.01.2006
(30)28.12.2001 DE 10164348
(54) Verfahren zur Herstellung von 1-Methoxy-2-propanol
(73)BASF Aktiengesellschaft
67056 Ludwigshafen (DE)
(72)Teles, Joaquim Henrique
Reiherstrasse 29a
67166 Otterstadt (DE)
(51) C07 F0017/00 (2006.01)
C07 F0007/28 (2006.01)
C08F0004/76 (2006.01)
C08F0012/08 (2006.01)
(11) 01 404 690
(21) 02751855.4
(11) 01 207 161
(51) C 07 D 0513/04 (2006.01) Z C 07 D 0491/048 (2006.01)
(11) 01 207 161
(51) C 07 D 0513/14 (2006.01) Z C 07 D 0491/048 (2006.01)
(11) 01 207 161
(51) C07 F0007/18 (2006.01)
C07 F0009/48 (2006.01)
C07 F0009/50 (2006.01)
C07 F0009/572 (2006.01)
C07 F0009/653 (2006.01)
C07 F0009/6547 (2006.01)
C07 F0009/6571 (2006.01)
C07 F0015/00 (2006.01)
(11) 01 097 158
(21) 99933785.0
(22)09.07.1999 (86)en
(43)09.05.2001(87)en
(24) 25.01.2006
(30)10.07.1998 US 113478
20.11.1998 US 196855
13.01.1999 US 231315
27.01.1999 US 239024
(54) LIGANDEN FÜR METALLE UND
METALL-KATALYSIERTES VERFAHREN
(73)MASSACHUSETTS INSTITUTE OF TECHNOLOGY
77 Massachusetts Avenue
Cambridge, MA 02139 (US)
(72)BUCHWALD, Stephen
25 Lancaster Road
Newton, MA 02158 (US)
OLD, David, W.
7 Adams Street No. 2
Somerville, MA 02145 (US)
WOLFE, John, P.
88 Berkeley AvenueNo. 16
Irvine CA 92612 (US)
PALUCKI, Michael
3 Horseshoe Drive
Belle Meade, NJ 08502 (US)
KAMIKAWA, Ken
1-14-19, Mozuumemachi
306,Sakai
Osaka 591-8032 (JP)
CHIEFFI, Andrew
Apt 25, 765 Somerville Avenue
Somerville, MA 02143 (US)
SINGER, Robert, A.
144 East 84th Street No.9D
New York, NY 10028 (US)
SADIGHI, Joseph, P.
Professor Joseph Sadighi MIT Department of Chemis
try MIT 18-390 Cambridge MA 02139 (US)
AHMAN, Jens
Cucumber Cottage, 25 Fisher Street
Sandwich, Kent CT 139 NJ (GB)
(86)PCT/US 1999/015450 (en)
(87)WO 2000/002887 20.1.2000
(51) C 07 F 0007/28 (2006.01) Z C 07 F 0017/00 (2006.01)
(11) 01 404 690
(51) C 07 F 0009/30 (2006.01) Z A 61 K 0031/44 (2006.01)
(11) 00 697 872
(51) C07 F0009/38 (2006.01)
(11) 01 423 397
(21) 02751375.3
(22)02.08.2002 (86)en
(43)02.06.2004(87)en
(24) 25.01.2006
(30)15.08.2001 GB 0119885
(54) VERFAHREN ZUR HERSTELLUNG VON
VINYLPHOSPHONSÄURE
(73)Rhodia Consumer Specialties Limited
Oak House, Reeds Crescent
Warford, Hertfordshire WD24 4QP (GB)
(72)JACKSON, Richard, David
The Fossil, Kinnersley, Severn Stoke
Worcestershire WR8 9JR (GB)
MATTHEWS, Kevin Roger Kenneth
212 Loxley Road, Staatford-upon-Avon
Warwickshire CV37 7DU (GB)
(86)PCT/GB 2002/003573 (en)
(87)WO 2003/016319 27.2.2003
(51) C 07 F 0009/38 (2006.01) Z A 61 K 0031/44 (2006.01)
201
31.1.2006 +pat+2
Commenti su questo manuale